| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | ctm | Design and biological evaluation of novel, balanced dual PPARa/g agonists | 3fei | 20 |
| 2 | ro7 | Aleglitazar, a new, potent, and balanced PPAR alpha/gamma agonist for the treatment of type II diabetes | 3g8i | 38 |
| 3 | 7ha | Crystal structure of peroxisome proliferator-activatedeceptor alpha (PPARalpha) complex with N-3-((2-(4-Chlorophenyl)-5-methyl-1,3-oxazol-4-yl)methoxy)benzyl)-N-(methoxycarbonyl)glycine | 3kdt | 260 |
| 4 | nks | Crystal structure of peroxisome proliferator-activatedeceptor alpha (PPARalpha) complex with N-3-((2-(4-Chlorophenyl)-5-methyl-1,3-oxazol-4-yl)methoxy)benzyl)-N-((4-methylphenoxy)carbonyl)glycine | 3kdu | 347 |
| 5 | az2 | CRYSTAL STRUCTURE OF THE LIGAND BINDING DOMAIN FROM HUMAN PPAR-ALPHA IN COMPLEX WITH THE AGONIST AZ 242 | 1i7g | 1000 |