| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 6xh | CREBBP bromodomain in complex with Cpd59 ((S)-1-(3-((2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)phenyl)amino)-1-(tetrahydrofuran-3-yl)-6,7-dihydro-1H-pyrazolo[4,3-c]pyridin-5(4H)-yl)ethanone) | 5ktx | 20 |
| 2 | 6xg | CREBBP bromodomain in complex with Cpd 44 (3-((5-acetyl-1-(cyclopropylmethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)amino)-N-isopropylbenzamide) | 5ktw | 30 |
| 3 | 69b | Crystal structure of the bromodomain of human CREBBP bound to the benzodiazepinone G02857790 | 5i89 | 33 |
| 4 | 6f9 | Crystal structure of the bromodomain of human CREBBP in complex with a benzoxazepine compound | 5j0d | 134 |
| 5 | 99e | Crystal structure of the human bromodomain of CREBBP bound to the inhibitor XDM-CBP | 5nu3 | 230 |
| 6 | 69a | Crystal structure of the bromodomain of human CREBBP bound to the benzodiazepinone G02778174 | 5i86 | 530 |
| 7 | 6xb | Crystal structure of the bromodomain of human CREBBP bound to pyrazolopiperidine scaffold | 5ktu | 620 |
| 8 | ul4 | Crystal structure of the bromodomain of human CREBBP in complex with UL04 | 4tqn | 770 |
| 9 | 77x | Structure of bromodomain of CREBBP with a pyrazolo[4,3-c]pyridin fragment | 5tb6 | 1530 |
| 10 | 68y | Crystal structure of the bromodomain of human CREBBP bound to the benzodiazepinone G02773986 | 5i83 | 4100 |
| 11 | xdm | Crystal structure of the bromodomain of human CREBBP bound to the inhibitor XDM1 | 5lpj | 1.01e+004 |
| 12 | 71x | Crystal structure of the bromodomain of human CREBBP bound to the inhibitor XDM3c | 5lpl | 1.2e+004 |