| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | mm3 | CRYSTAL STRUCTURE OF MMP3 COMPLEXED WITH A THIAZEPINE BASED INHIBITOR. | 1d5j | 0.7 |
| 2 | spc | CRYSTAL STRUCTURE OF MMP3 COMPLEXED WITH A MODIFIED PROLINE SCAFFOLD BASED INHIBITOR. | 1d7x | 3 |
| 3 | in7 | X-RAY STRUCTURE OF HUMAN STROMELYSIN CATALYTIC DOMAIN COMPLEXED WITH NON-PEPTIDE INHIBITORS: IMPLICATIONS FOR INHIBITOR SELECTIVITY | 1b8y | 14 |
| 4 | in9 | CRYSTAL STRUCTURE OF THE CATALYTIC DOMAIN OF HUMAN FIBROBLAST STROMELYSIN-1 INHIBITED WITH THIADIAZOLE INHIBITOR PNU-142372 | 1usn | 18 |
| 5 | n25 | DISCOVERY OF POTENT, ACHIRAL MATRIX METALLOPROTEINASE INHIBITORS | 1bqo | 18.4 |
| 6 | s80 | DESIGN AND SYNTHESIS OF CONFORMATIONALLY-CONSTRAINED MMP INHIBITORS | 1biw | 104 |
| 7 | hqq | X-ray Structure of a Novel Matrix Metalloproteinase Inhibitor Complexed to Stromelysin | 1g4k | 2000 |