| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 6dv | Crystal structure of stabilized A2A adenosine receptor A2AR-StaR2-bRIL in complex with compound 12x at 2.1A resolution | 5iub | 0.35 |
| 2 | zma | Crystal structure of stabilized A2A adenosine receptor A2AR-StaR2-bRIL in complex with ZM241385 at 1.7A resolution | 5iu4 | 0.53 |
| 3 | 6dy | Crystal structure of stabilized A2A adenosine receptor A2AR-StaR2-bRIL in complex with compound 12c at 1.9A resolution | 5iu7 | 1.1 |
| 4 | 6dx | Crystal structure of stabilized A2A adenosine receptor A2AR-StaR2-bRIL in complex with compound 12b at 2.2A resolution | 5iua | 1.5 |
| 5 | zma | The 2.6 A Crystal Structure of a Human A2A Adenosine Receptor bound to ZM241385. | 3eml | 1.8 |
| 6 | nec | Thermostabilised HUMAN A2a Receptor with NECA bound | 2ydv | 13.8 |
| 7 | 6dz | Crystal structure of stabilized A2A adenosine receptor A2AR-StaR2-bRIL in complex with compound 12f at 2.0A resolution | 5iu8 | 18 |
| 8 | adn | Thermostabilised HUMAN A2a Receptor with adenosine bound | 2ydo | 30.9 |