| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 4e1 | Crystal structure of DYRK1A in complex with 10-Iodo-substituted 11H-indolo[3,2-c]quinoline-6-carboxylic acid inhibitor 5j | 4ylj | 6 |
| 2 | 2c3 | The crystal structure of DYRK1a with a bound pyrido[2,3-d]pyrimidine inhibitor | 4mq1 | 12 |
| 3 | 2c4 | The crystal structure of DYRK1a with a bound pyrido[2,3-d]pyrimidine inhibitor | 4mq2 | 97 |
| 4 | ehb | human DYRK1A/inhibitor complex | 3anq | 180 |
| 5 | 4e2 | Crystal structure of DYRK1A in complex with 10-Chloro-substituted 11H-indolo[3,2-c]quinolone-6-carboxylic acid inhibitor 5s | 4ylk | 180 |