| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
|---|---|---|---|---|
| 1 | 4k7 | Crystal Structure of human phosphorylated IRE1alpha in complex with a type III kinase inhibitor (GSK2850163A) | 4yz9 | 20 |
| 2 | 4l5 | Crystal structure of human IRE1 cytoplasmic kinase-RNase region - complex with imidazopyridine compound 3 | 4z7h | 218 |