| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | yam | Crystal Structure Analysis of Focal Adhesion Kinase with a Methanesulfonamide Diaminopyrimidine Inhibitor | 3bz3 | 1.5 |
| 2 | bi9 | Focal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor | 2jkk | 6.24 |
| 3 | vg8 | Focal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor | 2jkq | 7.7 |
| 4 | bij | Focal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor | 2jko | 7.7 |
| 5 | bii | Focal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor | 2jkm | 17.76 |
| 6 | 10n | FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH N-{3-[(5-Cyano-2-phenyl-1H-pyrrolo[2,3-b]pyridin-4-ylamino)- methyl]-pyridin-2-yl}-N-methyl-methanesulfonamide | 4gu6 | 44 |
| 7 | 7py | Crystal Structure of Focal Adhesion Kinase Domain Complexed with 7H-Pyrrolo [2,3-d] pyrimidine Derivative | 2etm | 212 |
| 8 | kgw | Focal Adhesion Kinase catalytic domain in complex with a diarylamino- 1,3,5-triazine inhibitor | 4brx | 320 |
| 9 | 5ri | Focal Adhesion Kinase catalytic domain in complex with a diarylamino- 1,3,5-triazine inhibitor | 4c7t | 400 |
| 10 | 1bq | Structure of Focal Adhesion Kinase catalytic domain in complex with hinge binding pyrazolobenzothiazine compound. | 4i4e | 500 |
| 11 | kao | FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH 1-(5-tert-Butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-(4-pyridin-3- yl-phenyl)-urea | 4kao | 770 |
| 12 | 4gu | Focal adhesion kinase catalytic domain in complex with (2-Fluoro-phenyl)-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)-amine | 4gu9 | 4.3e+004 |