| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 66t | FGFR1 in complex with AZD4547. | 4v05 | 0.2 |
| 2 | 07j | Co-structure of Fibroblast Growth Factor Receptor 1 kinase domain with 3-(2,6-dichloro-3,5-dimethoxy-phenyl)-1-{6-[4-(4-ethyl-piperazin-1-yl)-phenylamino]-pyrimidin-4-yl}-1-methyl-urea (BGJ398) | 3tt0 | 0.9 |
| 3 | 66t | Crystal Structure of FGFR1 (C488A, C584S) in complex with AZD4547 (N-{3-[2-(3,5-DIMETHOXYPHENYL)ETHYL]-1H-PYRAZOL-5-YL}-4-[(3R,5S)-3,5-DIMETHYLPIPERAZIN-1-YL]BENZAMIDE) | 4rwj | 2 |
| 4 | 0s9 | Crystal structure of Human Fibroblast Growth Factor Receptor 1 Kinase domain in complex with compound 8 | 4f65 | 2.5 |
| 5 | 2k5 | Crystal structure of human fibroblast growth factor receptor 1 kinase domain in complex with pyrazolaminopyrimidine 1 | 4nk9 | 3.1 |
| 6 | xoj | FGFR1 ligand complex | 5a4c | 5.7 |
| 7 | 0li | FGFR1 in complex with ponatinib (co-crystallisation). | 4v01 | 7.7 |
| 8 | 0li | FGFR1 in complex with ponatinib. | 4v04 | 7.7 |
| 9 | 4ut | Crystal structure of FGFR1 kinase domain in complex with 7n | 4zsa | 15 |
| 10 | 38o | FGFR1 in complex with dovitinib | 5a46 | 22 |
| 11 | pd1 | CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FGF RECEPTOR 1 IN COMPLEX WITH INHIBITOR PD173074 | 2fgi | 45.2 |
| 12 | 0s8 | Crystal structure of Human Fibroblast Growth Factor Receptor 1 Kinase domain in complex with compound 6 | 4f64 | 63.1 |
| 13 | 66t | Crystal structure of V561M FGFR1 gatekeeper mutation (C488A, C584S, V561M) in complex with N-{3-[2-(3,5-DIMETHOXYPHENYL)ETHYL]-1H-PYRAZOL-5-YL}-4-[(3R,5S)-3,5-DIMETHYLPIPERAZIN-1-YL]BENZAMIDE (AZD4547) | 4rwk | 64 |
| 14 | 38o | FGFR1 mutant with an inhibitor | 5am7 | 64.5 |
| 15 | 2m2 | Crystal structure of human fibroblast growth factor receptor 1 kinase domain in complex with pyrazolaminopyrimidine 3 | 4nks | 67.9 |
| 16 | 38o | Native FGFR1 with an inhibitor | 5am6 | 185 |
| 17 | 2k7 | Crystal structure of human fibroblast growth factor receptor 1 kinase domain in complex with pyrazolaminopyrimidine 2 | 4nka | 311.4 |
| 18 | 0s7 | Crystal structure of Human Fibroblast Growth Factor Receptor 1 Kinase domain in complex with compound 1 | 4f63 | 500 |
| 19 | 3rh | Crystal structure of the catalytic domain of FGFR1 kinase in complex with ARQ 069 | 3rhx | 840 |
| 20 | c4f | FGFR TYROSINE KINASE DOMAIN IN COMPLEX WITH 3-(3-methoxybenzyl)-7-azaindole | 3c4f | 1900 |
| 21 | su1 | CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 IN COMPLEX WITH SU5402 INHIBITOR | 1fgi | 1e+004 |
| 22 | su2 | CRYSTAL STRUCTURE OF THE TYROSINE KINASE DOMAIN OF FIBROBLAST GROWTH FACTOR RECEPTOR 1 IN COMPLEX WITH SU4984 INHIBITOR | 1agw | 2e+004 |