| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 6lq | GSK3b in complex with inhibitor | 4acg | 0.22 |
| 2 | 2we | Structure of a carboxamide compound (3) (2-{2-[(CYCLOPROPYLCARBONYL)AMINO]PYRIDIN-4-YL}-4-OXO-4H-1LAMBDA~4~,3-THIAZOLE-5-CARBOXAMIDE) to GSK3b | 4ptc | 1.1 |
| 3 | z92 | 3-Aryl-4-(arylhydrazono)-1H-pyrazol-5-ones: Highly ligand efficient and potent inhibitors of GSK3 | 3l1s | 2 |
| 4 | 3uo | Crystal structure of GSK3b in complex with Compound 15: 2-[(cyclopropylcarbonyl)amino]-N-(4-methoxypyridin-3-yl)pyridine-4-carboxamide | 5f94 | 3.4 |
| 5 | gr9 | GSK3b in complex with inhibitor | 4acd | 4.9 |
| 6 | brw | GLYCOGEN SYNTHASE KINASE 3 BETA COMPLEXED WITH 6-BROMOINDIRUBIN-3'-OXIME | 1uv5 | 5 |
| 7 | 65c | Co-structure of human glycogen synthase kinase beta with a selective (5-imidazol-2-yl-4-phenylpyrimidin-2-yl)[2-(2-pyridylamino)ethyl]amine inhibitor | 6b8j | 5 |
| 8 | 2wg | Structure of a carboxamine compound (26) (2-{2-[(CYCLOPROPYLCARBONYL)AMINO]PYRIDIN-4-YL}-4-METHOXYPYRIMIDINE-5-CARBOXAMIDE) to GSK3b | 4ptg | 5.9 |
| 9 | z48 | Crystal structure of GSK3b in complex with a pyrimidylpyrrole inhibitor | 3i4b | 7 |
| 10 | 6qh | Crystal structure of GSK-3beta complexed with PF-04802367, a highly selective brain-penetrant kinase inhibitor | 5k5n | 9 |
| 11 | 3up | Crystal structure of GSK3b in complex with Compound 18: 2-[(cyclopropylcarbonyl)amino]-N-(4-phenylpyridin-3-yl)pyridine-4-carboxamide | 5f95 | 9.8 |
| 12 | 55e | 6-Amino-4-(pyrimidin-4-yl)pyridones: Novel Glycogen Synthase Kinase-3 Inhibitors | 3q3b | 17.2 |
| 13 | 7yg | GSK3b in complex with inhibitor | 4acc | 20 |
| 14 | kdi | GSK3b in complex with inhibitor | 4ach | 22 |
| 15 | tmu | crystal structure of Glycogen synthase kinase 3 in complexed with inhibitor | 1q5k | 38 |
| 16 | 679 | GSK-3 Beta complexed with Inhibitor I-5 | 1q4l | 40 |
| 17 | 65a | X-RAY CRYSTAL STRUCTURE OF GSK3B IN COMPLEX WITH BRD3937 | 5hlp | 54 |
| 18 | 2wf | Structure of a carvoxamide compound (15) (N-[4-(ISOQUINOLIN-7-YL)PYRIDIN-2-YL]CYCLOPROPANECARBOXAMIDE) to GSK3b | 4pte | 74 |
| 19 | zrm | Identification of 2-(4-pyridyl)thienopyridinones as GSK-3beta inhibitors | 3zrm | 130 |
| 20 | 553 | Crystal structure of GSK-3 beta in complex with NMS-869553A | 3du8 | 146 |
| 21 | sjj | 5-aryl-4-carboxamide-1,3-oxazoles: potent and selective GSK-3 inhibitors | 4afj | 398 |