| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | bd2 | Crystal structure of cAMP-dependent protein kinase complexed with balanol analog 2 | 1re8 | 0.3 |
| 2 | 4l7 | Protein Kinase A in complex with an Inhibitor | 4uja | 0.9 |
| 3 | s3n | Protein Kinase A in complex with an Inhibitor | 4uj9 | 2 |
| 4 | 796 | Discovery of 2-Pyrimidyl-5-Amidothiophenes as Novel and Potent Inhibitors for AKT: Synthesis and SAR Studies | 2gu8 | 2.6 |
| 5 | b1l | Crystal structure of cAMP-dependent protein kinase complexed with balanol analog 1 | 1rej | 5 |
| 6 | l20 | Structure of cAMP-dependent protein kinase complexed with A-443654 | 2jds | 6.3 |
| 7 | l9n | crystal structure of PKAB3 (pka triple mutant V123A, L173M, Q181K) with compound 27 | 3l9n | 8.6 |
| 8 | 8bq | Protein Kinase A in complex with an Inhibitor | 4ujb | 10 |
| 9 | r69 | Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants | 1xh9 | 17 |
| 10 | gvk | Structure of PKA-PKB chimera complexed with 6-(4-(4-(4-Chloro-phenyl) -piperidin-4-yl)-phenyl)-9H-purine | 2uw0 | 20 |
| 11 | gvn | Structure of PKA-PKB chimera complexed with (R)-2-(4-chloro-phenyl)- 2-(4-1H-pyrazol-4-yl)-phenyl)-ethylamine | 2uw5 | 31 |
| 12 | r69 | Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants | 1xh4 | 34 |
| 13 | r94 | Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants | 1xh6 | 48 |
| 14 | l9m | Crystal structure of PKAB3 (pka triple mutant V123A, L173M, Q181K) with compound 18 | 3l9m | 50 |
| 15 | nvv | Protein Kinase A in complex with an Inhibitor | 4uj2 | 80 |
| 16 | r96 | Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants | 1xh7 | 150 |
| 17 | l9l | Crystal structure of pka with compound 36 | 3l9l | 167 |
| 18 | b8l | Crystal structure of cAMP-dependent protein kinase complexed with balanol analog 8 | 1rek | 200 |
| 19 | gvo | Structure of PKA-PKB chimera complexed with (S)-2-(4-chloro-phenyl)- 2-(4-1H-pyrazol-4-yl)-phenyl)-ethylamine | 2uw6 | 280 |
| 20 | ske | Protein kinase A sixfold mutant model of Aurora B with inhibitor JNJ-7706621 | 3ama | 297 |
| 21 | nvx | Protein Kinase A in complex with an Inhibitor | 4uj1 | 300 |
| 22 | nu3 | PKA-S6K1 Chimera with compound 1 (NU1085) bound | 4c35 | 560 |
| 23 | vx6 | Protein kinase A sixfold mutant model of Aurora B with inhibitor VX-680 | 3amb | 660 |
| 24 | ss5 | PKA structures of indazole-pyridine series of AKT inhibitors | 2uzv | 1360 |
| 25 | nvx | PKAB3 in complex with pyrrolidine inhibitor 34a | 4z84 | 1500 |
| 26 | r55 | Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants | 1xh8 | 1700 |
| 27 | xfe | Human cyclic AMP-dependent protein kinase PKA inhibitor complex | 3mvj | 3200 |
| 28 | r68 | Crystal Structures of Protein Kinase B Selective Inhibitors in Complex with Protein Kinase A and Mutants | 1xh5 | 3400 |
| 29 | y27 | The Catalytic Subunit of cAMP-dependent Protein Kinase (PKA) in Complex with Rho-kinase Inhibitor Y-27632 | 1q8t | 1.75e+004 |
| 30 | gvq | Structure of PKA-PKB chimera complexed with 2-(4-chloro-phenyl)-2- phenyl-ethylamine | 2uw8 | 7.7e+004 |