| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
|---|---|---|---|---|
| 1 | 0li | Crystal structure of KIT in complex with ponatinib | 4u0i | 6 |
| 2 | b49 | KIT kinase domain in complex with sunitinib | 3g0e | 20 |
| 3 | b49 | KIT kinase domain mutant D816H in complex with sunitinib | 3g0f | 22 |
| 4 | sti | STRUCTURAL BASIS FOR THE AUTOINHIBITION AND STI-571 INHIBITION OF C-KIT TYROSINE KINASE | 1t46 | 370 |