| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 8gy | Structure-Based Design of ASK1 Inhibitors as Potential First-in-Class Agents for Heart Failure | 5uox | 5.01 |
| 2 | bh9 | Crystal Structures of Ask1-inhibitor Complexes | 4bhn | 6.31 |
| 3 | 8gv | Structure-Based Design of ASK1 Inhibitors as Potential First-in-Class Agents for Heart Failure | 5uor | 6.31 |
| 4 | ie8 | Crystal Structures of Ask1-inhibitor Complexes | 4bid | 7.94 |
| 5 | 8gs | Structure-Based Design of ASK1 Inhibitors as Potential First-in-Class Agents for Heart Failure | 5up3 | 12.59 |
| 6 | im6 | Crystal structure of human apoptosis signal-regulating kinase 1 (ASK1) with imidazopyridine inhibitor | 3vw6 | 14 |
| 7 | ieo | Crystal Structures of Ask1-inhibitor Complexes | 4bib | 250 |
| 8 | ie6 | Crystal Structures of Ask1-inhibitor Complexes | 4bie | 250 |
| 9 | 8v7 | Structure-based drug design of novel ASK1 inhibitors using a fully integrated lead optimization strategy | 5v24 | 400 |