| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
|---|---|---|---|---|
| 1 | rf4 | Crystal structure of PDK1 in complex with ATP and the PIF-pocket ligand RF4 | 4xx9 | 8400 |
| 2 | p47 | Crystal structure of Human PDK1 kinase domain in complex with an allosteric activator bound to the PIF-pocket | 3hrf | 1.03e+004 |