| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 4tw | ROCK 1 bound to a pyridine thiazole inhibitor | 5bml | 10 |
| 2 | 07r | Rho-associated protein kinase 1 (ROCK 1) IN COMPLEX WITH RKI1447 | 3twj | 14.5 |
| 3 | 3nc | X-Ray Co-structure of Rho-Associated Protein Kinase (ROCK1) with a potent 2H-isoquinolin-1-one inhibitor | 3ncz | 15 |
| 4 | 07q | Human Rho-associated protein kinase 1 (ROCK 1) in COMPLEX WITH RKI1342 | 3tv7 | 30 |
| 5 | 3j7 | Crystal Structure of ROCK 1 bound to YB-15-QD37 | 4w7p | 32 |
| 6 | y27 | Crystal Structure of ROCK I bound to Y-27632 | 2etr | 150 |
| 7 | hfs | Crystal Structure of ROCK 1 bound to hydroxyfasudil | 2etk | 150 |