The Ligandable Human Proteome

Home

Angiopoietin-1 receptor

Protein kinase domain

IndexLigand NameStructurePDB codeCompound Potency nM
1rajSynthesis, Structural Analysis, and SAR Studies of Triazine Derivatives as Potent, Selective Tie-2 Inhibitors2oo81
2mr9Evolution of a highly Selective and Potent 2-(Pyridin-2-yl)-1,3,5-triazine Tie-2 Kinase Inhibitor2p4i10
3muhSynthesis, Structural Analysis, and SAR Studies of Triazine Derivatives as Potent, Selective Tie-2 Inhibitors2osc17
4qq1Structure of the Tie2 kinase domain in complex with a thiazolopyrimidine inhibitor2wqb540