| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 96m | Crystal structure of human WEE1 kinase domain in complex with PD-166285 | 5vc5 | 11 |
| 2 | 8x7 | CRYSTAL STRUCTURE OF HUMAN WEE1 KINASE DOMAIN IN COMPLEX WITH MK1775 | 5v5y | 13.4 |
| 3 | p48 | crystal structure of human WEE1 kinase domain in complex with PHA-848125 | 5vc6 | 13.6 |
| 4 | 396 | Wee1 kinase complex with inhibitor PD352396 | 3bi6 | 15 |
| 5 | xzn | Crystal structure of HUMAN WEE1 KINASE domain in complex with Bosutinib-isomer | 5vc4 | 43.7 |
| 6 | 61e | Wee1 kinase complex with inhibitor PD331618 | 3biz | 58 |
| 7 | db8 | CRYSTAL STRUCTURE OF HUMAN WEE1 KINASE DOMAIN IN COMPLEX WITH BOSUTINIB | 5vc3 | 77.5 |
| 8 | 34w | crystal structure of human WEE1 kinase domain in complex with PF-03814735 | 5vd2 | 78.7 |