| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | i96 | Human Methionine Aminopeptidase-2 Complexed with SB-587094 | 2oaz | 2 |
| 2 | f77 | h-MetAP2 complexed with A773812 | 2ea2 | 16 |
| 3 | ao1 | Crystal Structure of MetAP2 complexed with A311263 | 1r5g | 30 |
| 4 | 7bf | CRYSTAL STRUCTURE OF HUMAN METHIONINE AMINOPEPTIDASE-2 IN COMPLEX; WITH AN INHIBITOR 5-((R)-1-[1,2,4]Triazolo[1,5-a]pyrimidin-7-yl-pyrrolidin-2-ylmethoxy)-isoquinoline | 5lyx | 38 |
| 5 | f79 | h-MetAP2 complexed with A797859 | 2ea4 | 46 |
| 6 | ao5 | Crystal Structure of MetAP2 complexed with A357300 | 1r58 | 110 |
| 7 | ao2 | Crystal Structure of MetAP2 complexed with A320282 | 1r5h | 180 |
| 8 | 52t | Structure of human methionine aminopeptidase-2 complexed with spiroepoxytriazole inhibitor (+)-31a | 5cls | 220 |
| 9 | 7bh | CRYSTAL STRUCTURE OF HUMAN METHIONINE AMINOPEPTIDASE-2 IN COMPLEX; WITH AN INHIBITOR 6-((R)-2-o-Tolyloxymethyl-pyrrolidin-1-yl)-9H-purine | 5lyw | 700 |
| 10 | 57r | Structure of human methionine aminopeptidase-2 complexed with spiroepoxytriazole inhibitor (+)-31b | 5d6f | 4.3e+004 |
| 11 | 94a | Structure of human methionine aminopeptidase 2 with covalent spiroepoxytriazole inhibitor (-)-31b | 5d6e | 5e+004 |