| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 7l6 | Structure of human GLP SET-domain (EHMT1) in complex with inhibitor MS0124 | 5tuz | 40 |
| 2 | 9hj | Structure of human GLP SET-domain (EHMT1) in complex with inhibitor 13 | 5vsd | 57 |
| 3 | 9hg | Structure of human GLP SET-domain (EHMT1) in complex with inhibitor 17 | 5vsf | 94 |
| 4 | e72 | Human G9a-like (GLP, also known as EHMT1) in complex with inhibitor E72 | 3mo5 | 136 |
| 5 | e11 | Human G9a-like (GLP, also known as EHMT1) in complex with inhibitor E11 | 3mo0 | 154 |
| 6 | e67 | human G9a-like (GLP, also known as EHMT1) in complex with inhibitor E67 | 3mo2 | 244 |
| 7 | q4a | G9a-like protein lysine methyltransferase inhibition by BIX-01294 | 3fpd | 700 |