| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | kpk | Crystal Structure of the human Chymase with TJK002 | 4kp0 | 2.24 |
| 2 | 8w3 | Human chymase in complex with 7-oxo-3-(phenoxyimino)-1,4-diazepane derivative | 5yjm | 21 |
| 3 | 1p9 | Crystal Structure of Human Chymase in Complex with Fragment Linked Benzimidazolone Inhibitor: (3S)-3-{3-[(6-bromo-2-oxo-2,3-dihydro-1H-indol-4-yl)methyl]-2-oxo-2,3-dihydro-1H-benzimidazol-1-yl}hexanoic acid | 4k69 | 40 |
| 4 | 0bb | Crystal Structure of Human Chymase with Benzimidazolone Inhibitor | 3s0n | 180 |
| 5 | 8w6 | Human chymase in complex with 3-(ethoxyimino)-7-oxo-1,4-diazepane derivative | 5yjp | 240 |