| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | ntx | Crystal structure of matriptase in complex with inhibitor | 4o97 | 3 |
| 2 | nt4 | Crystal structure of matriptase in complex with inhibitor | 4o9v | 10 |
| 3 | n4c | Crystal Structure of Matriptase in complex with Inhibitor"". | 4jzi | 40 |
| 4 | n4a | Crystal Structure of Matriptase in complex with Inhibitor | 4jyt | 40 |
| 5 | 730 | Crystal Structure of Matriptase with Inhibitor CJ-730 | 2gv6 | 46 |
| 6 | f4d | Crystal Structure of Matriptase in complex with Inhibitor | 4jz1 | 200 |
| 7 | 3km | CRYSTAL STRUCTURE of MATRIPTASE in COMPLEX WITH INHIBITOR | 4r0i | 300 |