The Ligandable Human Proteome

Home

Bromodomain-containing protein 9

Bromodomain

IndexLigand NameStructurePDB codeCompound Potency nM
1tvuBROMODOMAIN OF HUMAN BRD9 WITH 7-(3,4-dimethoxyphenyl)-N-(1,1-dioxo-1- thian-4-yl)-5-methyl-4-oxo-4H,5H-thieno-3,2-c-pyridine-2-carboxamide4uiu12.6
25u6Crystal structure of the BRD9 bromodamian in complex with BI-9564.5f1h14.1
35swCRYSTAL STRUCTURE OF BRD9 IN COMPLEX WITH BI-72735eu115.4
4xzbBROMODOMAIN OF HUMAN BRD9 WITH N-(1,1-dioxo-1-thian-4-yl)-5-methyl-4- oxo-7-3-(trifluoromethyl)phenyl-4H,5H-thieno-3,2-c-pyridine-2- carboximidamide4uiv15.8
55u2Crystal structure of the bromodomain of BRD9 in complex with compound 9.5f1l21
6bmfCrystal structure of the bromodomain of human BRD9 in complex with bromosporine (BSP)5igm41.7
7h1bBROMODOMAIN OF HUMAN BRD9 WITH N-(1,1-dioxo-1-thian-4-yl)-5-ethyl-4- oxo-7-3-(trifluoromethyl)phenyl-4H,5H-thieno-3,2-c-pyridine-2- carboximidamide4uiw50
869gBRD9 in complex with Cpd4 ((E)-3-(6-(but-2-en-1-yl)-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)-N,N-dimethylbenzamide)5i7y52
9n1dBROMODOMAIN OF HUMAN BRD9 WITH 7-(3,4-dimethoxyphenyl)-2-(4- methanesulfonylpiperazine-1-carbonyl)-5-methyl-4H,5H-thieno-3,2-c- pyridin-4-one4uit200
105tyCrystal structure of the BRD9 bromodomain in complex with compound 3.5f2p3.75e+004