| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
|---|---|---|---|---|
| 1 | 99e | Crystal structure of the human bromodomain of EP300 bound to the inhibitor XDM-CBP | 5nu5 | 470 |
| 2 | 71y | Crystal structure of the bromodomain of human Ep300 bound to the inhibitor XDM3d | 5lpm | 2770 |
| 3 | xdm | Crystal structure of the bromodomain of human EP300 bound to the inhibitor XDM1 | 5lpk | 3060 |