| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | mkr | Crystal Structure of KSP in complex with Inhibitor 1 | 2q2y | 1.6 |
| 2 | n4t | crystal structure of KSP in complex with inhibitor 19 | 2fl2 | 2 |
| 3 | mkk | Crystal Structure of KSP in Complex with Inhibitor 22 | 2q2z | 2 |
| 4 | k30 | Crystal structure of KSP in complex with inhibitor 30 | 3cjo | 2.2 |
| 5 | n2t | crystal structure of KSP in complex with inhibitor 13 | 2fky | 2.6 |
| 6 | emq | X-ray structure of mitotic kinesin-5 (KSP, KIF11, Eg5)in complex with the hexahydro-2H-pyrano[3,2-c]quinoline EMD 534085 | 3l9h | 8 |
| 7 | g7x | The mitotic kinesin Eg5 in complex with Mg-ADP and ispinesib | 4ap0 | 10 |
| 8 | 6lx | Eg5(WT) complex | 4bxn | 10 |
| 9 | n5t | crystal structure of KSP in complex with inhibitor 6 | 2fl6 | 38 |
| 10 | n9h | crystal structure of KSP in complex with inhibitor 9h | 2g1q | 44 |
| 11 | 2az | Crystal structure of the mitotic kinesin eg5 in complex with mg-adp and n-(3-aminopropyl)-n-((3-benzyl-5-chloro-4-oxo-3,4-dihydropyrrolo[2,1-f][1,2,4]triazin-2-yl)(cyclopropyl)methyl)-4-methylbenzamide | 2gm1 | 100 |
| 12 | 3qc | Crystal structure of the mitotic kinesin eg5 (ksp) in complex with mg-adp and (r)-4-(3-hydroxyphenyl)-n,n,7,8-tetramethyl-3,4-dihydroisoquinoline-2(1h)-carboxamide | 2fme | 104 |
| 13 | moy | Crystal structure of human kinesin Eg5 in complex with (R)-mon97, a new monastrol-based inhibitor that binds as (R)-enantiomer | 2ieh | 110 |
| 14 | egb | Crystal structure of human kinesin Eg5 in complex with (S)-dimethylenastron | 2x7d | 200 |
| 15 | l31 | Co-crystal structure of the human kinesin Eg5 with a novel tetrahydro-beta-carboline | 3k3b | 200 |
| 16 | l47 | Crystal structure of KSP in complex with inhibitor 1 | 1yrs | 450 |
| 17 | k02 | Crystal structure of KSP in complex with ADP and thiophene containing inhibitor 33 | 2uyi | 480 |
| 18 | k01 | Crystal structure of KSP in complex with ADP and thiophene containing inhibitor 15 | 2pg2 | 1700 |
| 19 | kz9 | Crystal structure of human kinesin Eg5 in complex with (S)-enastron | 2x7c | 2000 |
| 20 | k03 | Crystal structure of KSP in complex with ADP and thiophene containing inhibitor 37 | 2uym | 3100 |
| 21 | nat | Crystal structure of the motor protein KSP in complex with ADP and monastrol | 1q0b | 6700 |