| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | dwx | Crystal Structure of Autotaxin in Complex with 3BoA | 3wax | 13 |
| 2 | 7nb | Novel Imidazo[1,2-a]pyridine Derivatives with Potent Autotaxin/ENPP2 Inhibitor Activity | 5mhp | 15 |
| 3 | 4o3 | Structural basis for inhibition of human autotaxin by four novel compounds | 4zga | 20 |
| 4 | dwy | Crystal Structure of Autotaxin in Complex with 4BoA | 3way | 22 |
| 5 | dwv | Crystal Structure of Autotaxin in Complex with Compound 10 | 3wav | 180 |
| 6 | 7hr | Novel Imidazo[1,2-a]pyridine Derivatives with Potent Autotaxin/ENPP2 Inhibitor Activity | 5m7m | 357 |
| 7 | 4ny | Structural basis for inhibition of human autotaxin by four novel compounds | 4zg6 | 472 |
| 8 | dww | Crystal Structure of Autotaxin in Complex with 2BoA | 3waw | 580 |