| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | l6i | Structure of the Keap1 Kelch domain in complex with a small molecule inhibitor. | 5fnu | 1.3 |
| 2 | 0pl | Structure of the Keap1 Kelch domain in complex with a small molecule inhibitor. | 5fnt | 670 |
| 3 | 1vx | Structure of keap1 kelch domain with (1S,2R)-2-{[(1S)-5-methyl-1-[(1-oxo-1,3-dihydro-2H-isoindol-2-yl)methyl]-3,4-dihydroisoquinolin-2(1H)-yl]carbonyl}cyclohexanecarboxylic acid | 4l7d | 750 |
| 4 | 2fs | STRUCTURE OF KEAP1 KELCH DOMAIN WITH(1S,2R)-2-[(1S)-1-[(1-oxo-2,3-dihydro-1H-isoindol-2-Yl)methyl]-1,2,3,4-tetrahydroisoquinoline-2-Carbonyl]cyclohexane-1-carboxylic acid | 4n1b | 1100 |
| 5 | xyy | Structure of the Keap1 Kelch domain in complex with a small molecule inhibitor. | 5fns | 4000 |
| 6 | 1vw | Structure of keap1 kelch domain with 2-{[(1S)-2-{[(1R,2S)-2-(1H-tetrazol-5-yl)cyclohexyl]carbonyl}-1,2,3,4-tetrahydroisoquinolin-1-yl]methyl}-1H-isoindole-1,3(2H)-dione | 4l7c | 7400 |
| 7 | xms | Structure of the Keap1 Kelch domain in complex with a small molecule inhibitor. | 5fnr | 5.9e+004 |