| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | jb7 | Crystal Structure of Glutamate Carboxypeptidase II in a complex with urea-based inhibitor | 4ngm | 0.0449 |
| 2 | okd | Human glutamate carboxypeptidase II in complex with ARM-M4, urea- based inhibitor | 2xej | 1.34 |
| 3 | 2qq | X-ray structure of of human glutamate carboxypeptidase II (GCPII) in a complex with CEIBzL, a urea-based inhibitor N~2~-{[(1S)-1-carboxybut-3-yn-1-yl]carbamoyl}-N~6~-(4-iodobenzoyl)-L-lysine | 4oc2 | 5.3 |
| 4 | yze | Crystal structure of human glutamate carboxypeptidase II (GCPII) in a complex with DBIBzL, a urea-based inhibitor | 3iww | 11 |
| 5 | jrg | X-ray structure of human glutamate carboxypeptidase II in complex with a urea-based inhibitor (A25) | 3sjf | 23 |
| 6 | 5pu | X-ray structure of human glutamate carboxypeptidase II (GCPII) in complex with a hydroxamate inhibitor JHU242 | 5ely | 44 |
| 7 | 5q1 | X-ray structure of human glutamate carboxypeptidase II (GCPII) in complex with a hydroxamate inhibitor JHU241 | 5d29 | 97 |
| 8 | 2qn | X-ray structure of of human glutamate carboxypeptidase II (GCPII) in a complex with CPIBzL, a urea-based inhibitor N~2~-{[(1S)-1-carboxy-2-(pyridin-4-yl)ethyl]carbamoyl}-N~6~-(4-iodobenzoyl)-L-lysine | 4oc4 | 105 |
| 9 | 2r7 | X-ray structure of of human glutamate carboxypeptidase II (GCPII) in a complex with CCIBzL, a urea-based inhibitor N~2~-[(1-carboxycyclopropyl)carbamoyl]-N~6~-(4-iodobenzoyl)-L-lysine | 4oc0 | 318 |