Index | Ligand Name | Structure | PDB code | Compound Potency nM |
1 | 92o | Structure of the p53 cancer mutant Y220C with bound small molecule 7- ethyl-3-(piperidin-4-yl)-1H-indole | 5ab9 | 470 |
2 | p96 | Structure of the p53 core domain mutant Y220C bound to the stabilizing small molecule PhiKan5196 | 4agq | 9700 |
3 | p74 | Structure of the p53 core domain mutant Y220C bound to the stabilizing small molecule PhiKan5174 | 4ago | 1.55e+004 |
4 | p51 | Structure of the p53 core domain mutant Y220C bound to the stabilizing small molecule PhiKan5176 | 4agp | 2.06e+004 |
5 | y0v | Structure of the p53 cancer mutant Y220C in complex with 2-hydroxy-3, 5-diiodo-4-(1H-pyrrol-1-yl)benzoic acid | 5aoj | 2.1e+004 |
6 | p86 | Structure of the p53 core domain mutant Y220C bound to the stabilizing small molecule PhiKan5086 | 4agm | 1.05e+005 |
7 | nxg | Structure of the p53 core domain mutant Y220C bound to the stabilizing small molecule PhiKan5116 | 4agn | 1.07e+005 |
8 | p84 | Structure of the p53 core domain mutant Y220C bound to the stabilizing small molecule PhiKan784 | 4agl | 2.25e+005 |
9 | kmn | Structure of the p53 cancer Y220C bound to the stabilizing small molecule PhiKan5211 | 5a7b | 2.71e+005 |
10 | ul7 | Structure of the p53 cancer mutant Y220C with bound small-molecule stabilizer PhiKan5149 | 5aba | 1.04e+006 |
11 | fy8 | Structure of the p53 cancer mutant Y220C with bound small molecule PhiKan883 | 5aom | 1.27e+006 |