| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
|---|---|---|---|---|
| 1 | ku8 | Human poly(ADP-ribose) polymerase 3, catalytic fragment in complex with an inhibitor KU0058948 | 3c49 | 70 |
| 2 | 1va | Human artd3 (parp3) - catalytic domain in complex with inhibitor ME0368 | 4l7l | 1000 |
| 3 | 1vc | Human artd3 (parp3) - catalytic domain in complex with inhibitor ME0398 | 4l7u | 2200 |
| 4 | m00 | Human artd3 (parp3) - catalytic domain in complex with inhibitor ME0400 | 4l7r | 9600 |
| 5 | 1vb | Human artd3 (parp3) - catalytic domain in complex with inhibitor STO1542 | 4l7n | 1.44e+004 |