| Index | Ligand Name | Ligand Structure | Gene Name Primary | Protein Name | Uniprot ID | Gene Name Synonym | PDB Codes |
| 1 | os3 | | MTAP | S-methyl-5'-thioadenosine phosphorylase | Q13126 | MSAP | 6dz0 |
| 2 | os2 | | MTAP | S-methyl-5'-thioadenosine phosphorylase | Q13126 | MSAP | 6dyz |
| 3 | fmc | | MTAP | S-methyl-5'-thioadenosine phosphorylase | Q13126 | MSAP | 1sd1 |
| 4 | 7a6 | | MTAP | S-methyl-5'-thioadenosine phosphorylase | Q13126 | MSAP | 5tc6 |
| 5 | 5s7 | | MTAP | S-methyl-5'-thioadenosine phosphorylase | Q13126 | MSAP | 5eub |
| 6 | mta | | MTAP | S-methyl-5'-thioadenosine phosphorylase | Q13126 | MSAP | 1cg6 |
| 7 | tdi | | MTAP | S-methyl-5'-thioadenosine phosphorylase | Q13126 | MSAP | 5tc8 |
| 8 | mth | | MTAP | S-methyl-5'-thioadenosine phosphorylase | Q13126 | MSAP | 1sd2, 5tc7 |
| 9 | 4ct | | MTAP | S-methyl-5'-thioadenosine phosphorylase | Q13126 | MSAP | 3ozc, 3ozd |
| 10 | imh | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 1pf7, 1rr6, 1rt9, 2oc4, 2oc9, 2on6, 2q7o |
| 11 | im5 | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 3phb, 5ugf |
| 12 | gmp | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 1rfg |
| 13 | 22a | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 3k8q |
| 14 | 2fd | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 3ggs |
| 15 | dih | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 1rsz, 2a0w, 2a0x, 2a0y, 3bgs |
| 16 | msg | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 1yry |
| 17 | 3dg | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 1v45 |
| 18 | 2di | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 1v3q |
| 19 | nos | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 1rct |
| 20 | ac2 | | PNPH | Purine nucleoside phosphorylase | P00491 | NP | 1pwy |
| 21 | bau | | UPP2 | Uridine phosphorylase 2 | O95045 | | 3p0e, 3p0f |