| Index | Ligand Name | Ligand Structure | Gene Name Primary | Protein Name | Uniprot ID | Gene Name Synonym | PDB Codes |
| 1 | tst | | FKB1A | Peptidyl-prolyl cis-trans isomerase FKBP1A | P62942 | FKBP1 FKBP12 | 1j4i |
| 2 | sbx | | FKB1A | Peptidyl-prolyl cis-trans isomerase FKBP1A | P62942 | FKBP1 FKBP12 | 1fkh |
| 3 | sb3 | | FKB1A | Peptidyl-prolyl cis-trans isomerase FKBP1A | P62942 | FKBP1 FKBP12 | 1fkg |
| 4 | i63 | | FKBP4,FKBP5 | Peptidyl-prolyl cis-trans isomerase FKBP5 | Q13451 | AIG6 FKBP51 | 4drk, 4lay |
| 5 | jfk | | FKBP5 | Peptidyl-prolyl cis-trans isomerase FKBP5 | Q13451 | AIG6 FKBP51 | 4jfk |
| 6 | 5bh | | FKBP5 | Peptidyl-prolyl cis-trans isomerase FKBP5 | Q13451 | AIG6 FKBP51 | 5div |
| 7 | 3jp | | FKBP5 | Peptidyl-prolyl cis-trans isomerase FKBP5 | Q13451 | AIG6 FKBP51 | 4w9q |
| 8 | 1kz | | FKBP5 | Peptidyl-prolyl cis-trans isomerase FKBP5 | Q13451 | AIG6 FKBP51 | 4jfm |
| 9 | 1ky | | FKBP5 | Peptidyl-prolyl cis-trans isomerase FKBP5 | Q13451 | AIG6 FKBP51 | 4jfl |
| 10 | 1ku | | FKBP5 | Peptidyl-prolyl cis-trans isomerase FKBP5 | Q13451 | AIG6 FKBP51 | 4jfj |
| 11 | 1kt | | FKBP5 | Peptidyl-prolyl cis-trans isomerase FKBP5 | Q13451 | AIG6 FKBP51 | 4jfi |
| 12 | 384 | | FKBP5 | Peptidyl-prolyl cis-trans isomerase FKBP5 | Q13451 | AIG6 FKBP51 | 4tx0 |
| 13 | 9qn | | FKBP5 | Peptidyl-prolyl cis-trans isomerase FKBP5 | Q13451 | AIG6 FKBP51 | 5obk |