| Index | Ligand Name | Ligand Structure | Gene Name Primary | Protein Name | Uniprot ID | Gene Name Synonym | PDB Codes |
| 1 | jdg | | EHMT1 | Histone-lysine N-methyltransferase EHMT1 | Q9H9B1 | EUHMTASE1 GLP KIAA1876 KMT1D | 6mbo, 6mbp |
| 2 | e72 | | EHMT1 | Histone-lysine N-methyltransferase EHMT1 | Q9H9B1 | EUHMTASE1 GLP KIAA1876 KMT1D | 3mo5 |
| 3 | e67 | | EHMT1 | Histone-lysine N-methyltransferase EHMT1 | Q9H9B1 | EUHMTASE1 GLP KIAA1876 KMT1D | 3mo2 |
| 4 | q4a | | EHMT1 | Histone-lysine N-methyltransferase EHMT1 | Q9H9B1 | EUHMTASE1 GLP KIAA1876 KMT1D | 3fpd |
| 5 | e11 | | EHMT1 | Histone-lysine N-methyltransferase EHMT1 | Q9H9B1 | EUHMTASE1 GLP KIAA1876 KMT1D | 3mo0 |
| 6 | 90p | | EHMT1,EHMT2 | Histone-lysine N-methyltransferase EHMT2 | Q96KQ7 | BAT8 C6orf30 G9A KMT1C NG36 | 5v9i, 5v9j |
| 7 | 7kz | | EHMT1,EHMT2 | Histone-lysine N-methyltransferase EHMT1 | Q9H9B1 | EUHMTASE1 GLP KIAA1876 KMT1D | 5ttf, 5ttg |
| 8 | 7l6 | | EHMT1,EHMT2 | Histone-lysine N-methyltransferase EHMT1 | Q9H9B1 | EUHMTASE1 GLP KIAA1876 KMT1D | 5tuy, 5tuz |
| 9 | 9hj | | EHMT1,EHMT2 | Histone-lysine N-methyltransferase EHMT1 | Q9H9B1 | EUHMTASE1 GLP KIAA1876 KMT1D | 5vsc, 5vsd |
| 10 | 9hg | | EHMT1,EHMT2 | Histone-lysine N-methyltransferase EHMT1 | Q9H9B1 | EUHMTASE1 GLP KIAA1876 KMT1D | 5vse, 5vsf |
| 11 | ciq | | EHMT2 | Histone-lysine N-methyltransferase EHMT2 | Q96KQ7 | BAT8 C6orf30 G9A KMT1C NG36 | 3rjw |
| 12 | dxq | | EHMT2 | Histone-lysine N-methyltransferase EHMT2 | Q96KQ7 | BAT8 C6orf30 G9A KMT1C NG36 | 3k5k |
| 13 | 2od | | EHMT2 | Histone-lysine N-methyltransferase EHMT2 | Q96KQ7 | BAT8 C6orf30 G9A KMT1C NG36 | 4nvq |
| 14 | 75p | | KMT5A | N-lysine methyltransferase KMT5A | Q9NQR1 | PRSET7 SET07 SET8 SETD8 | 5t5g |
| 15 | 539 | | KMT5B | Histone-lysine N-methyltransferase KMT5B | Q4FZB7 | SUV420H1 | 5cpr |
| 16 | ks7 | | PRDM9 | Histone-lysine N-methyltransferase PRDM9 | Q9NQV7 | PFM6 | 6nm4 |
| 17 | 0n6 | | SETD7 | Histone-lysine N-methyltransferase SETD7 | Q8WTS6 | KIAA1717 KMT7 SET7 SET9 | 4e47 |
| 18 | ew4 | | SMYD2 | N-lysine methyltransferase SMYD2 | Q9NRG4 | KMT3C | 6cby |
| 19 | a4m | | SMYD2 | N-lysine methyltransferase SMYD2 | Q9NRG4 | KMT3C | 5wcg |
| 20 | ew1 | | SMYD2 | N-lysine methyltransferase SMYD2 | Q9NRG4 | KMT3C | 6cbx |
| 21 | nm4 | | SUV92 | Histone-lysine N-methyltransferase SUV39H2 | Q9H5I1 | KMT1B | 6p0r |