| Index | Ligand Name | Ligand Structure | Gene Name Primary | Protein Name | Uniprot ID | Gene Name Synonym | PDB Codes |
| 1 | 4i5 | | SIR1,SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 4i5i, 5d7q |
| 2 | 1ns | | SIR1,SIR3 | NAD-dependent protein deacetylase sirtuin-3, mitochondrial | Q9NTG7 | SIR2L3 | 4jt9, 4zzi |
| 3 | l5c | | SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 5yqo |
| 4 | l55 | | SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 5yqn |
| 5 | a2x | | SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 5yqm |
| 6 | 8k9 | | SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 5y0z |
| 7 | 7kj | | SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 5mat |
| 8 | 5gr | | SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 5dy5 |
| 9 | 5gn | | SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 5dy4 |
| 10 | 3te | | SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 4rmg, 4rmh |
| 11 | 3tk | | SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 4rmi |
| 12 | 8no | | SIR2 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 5y5n |
| 13 | ocz | | SIR2,SIR3 | NAD-dependent protein deacetylase sirtuin-2 | Q8IXJ6 | SIR2L SIR2L2 | 4bv3, 4bvb, 4bvh, 5d7p |
| 14 | 1nq | | SIR3 | NAD-dependent protein deacetylase sirtuin-3, mitochondrial | Q9NTG7 | SIR2L3 | 4jsr |
| 15 | 1nr | | SIR3 | NAD-dependent protein deacetylase sirtuin-3, mitochondrial | Q9NTG7 | SIR2L3 | 4jt8 |
| 16 | 7n2 | | SIR6 | NAD-dependent protein deacetylase sirtuin-6 | Q8N6T7 | SIR2L6 | 5mgn |
| 17 | 7m2 | | SIR6 | NAD-dependent protein deacetylase sirtuin-6 | Q8N6T7 | SIR2L6 | 5mf6 |