| Index | Gene Name Primary | Protein Name | Uniprot ID | Gene Name Synonym | Ligand Name | Structure | PDB Code | ligand desolvation | Ligand Structure | Compound Affinity nM |
| 1 | ACE | Angiotensin-converting enzyme | P12821 | DCP DCP1 | ft8 | Crystal structure of human Angiotensin-1 converting enzyme N-domain in complex with Omapatrilat. | 6h5x | 84.35 | | no data |
| 2 | ACE | Angiotensin-converting enzyme | P12821 | DCP DCP1 | lpr | Structure of human somatic angiontensin-I converting enzyme N domain with lisinopril | 2c6n | 70.17 | | 131.5 |
| 3 | ACE | Angiotensin-converting enzyme | P12821 | DCP DCP1 | eal | Complex of the anti-hypertensive drug enalaprilat and the human testicular angiotensin I-converting enzyme | 1uze | 75.31 | | 1.27 |
| 4 | ACE | Angiotensin-converting enzyme | P12821 | DCP DCP1 | lpr | Crystal Structure of Human Angiotensin Converting Enzyme in complex with lisinopril. | 1o86 | 75.24 | | 0.27 |
| 5 | ACE2 | Angiotensin-converting enzyme 2 | Q9BYF1 | | xx5 | Inhibitor Bound Human Angiotensin Converting Enzyme-Related Carboxypeptidase (ACE2) | 1r4l | 84.34 | | no data |