| Index | Gene Name | Protein Name | Drugs | PDB Code |
| 1 | 5HT2A | 5-hydroxytryptamine receptor 2A | Zotepine,Cholesterol | 6a94, 6a93 |
| 2 | PAR1 | Proteinase-activated receptor 1 | Vorapaxar | 3vw7 |
| 3 | PE2R3 | Prostaglandin E2 receptor EP3 subtype | Dinoprostone,Alprostadil | 6ak3 |
| 4 | CCR5 | C-C chemokine receptor type 5 | Maraviroc | 4mbs |
| 5 | ADRB2 | Beta-2 adrenergic receptor | Salmeterol,Timolol | 6mxt, 3d4s |
| 6 | MTR1A | Melatonin receptor type 1A | Ramelteon | 6me2 |
| 7 | NK1R | Substance-P receptor | Netupitant | 6hlp |
| 8 | 5HT2B | 5-hydroxytryptamine receptor 2B | Ergotamine,Methylergometrine,Ergometrine | 4ib4, 5tud, 4nc3, 6dry |
| 9 | 5HT1B | 5-hydroxytryptamine receptor 1B | Ergotamine,Dihydroergotamine | 4iar, 4iaq |
| 10 | 5HT2C | 5-hydroxytryptamine receptor 2C | Ergotamine | 6bqg |
| 11 | P2Y12 | P2Y purinoceptor 12 | Cholesterol | 4pxz, 4ntj |
| 12 | CNR1 | Cannabinoid receptor 1 | Cholesterol | 5xra, 5xr8, 6n4b |
| 13 | OPRM | Mu-type opioid receptor | Cholesterol | 5c1m, 4dkl |
| 14 | CCR9 | C-C chemokine receptor type 9 | Cholesterol | 5lwe |
| 15 | P2RY1 | P2Y purinoceptor 1 | Cholesterol | 4xnv |
| 16 | TA2R | Thromboxane A2 receptor | Cholesterol | 6iiv, 6iiu |
| 17 | AA2AR | Adenosine receptor A2a | Cholesterol | 5nlx |
| 18 | ACM2 | Muscarinic acetylcholine receptor M2 | Methscopolamine bromide, Scopolamine, Methscopolamine | 5yc8, 5zk8, 5zkc |
| 19 | AGTR1 | Type-1 angiotensin II receptor | Olmesartan | 4zud |
| 20 | ACM3 | Muscarinic acetylcholine receptor M3 | Tiotropium | 4u15 |
| 21 | ACM4 | Muscarinic acetylcholine receptor M4 | Tiotropium | 5dsg |
| 22 | ACM1 | Muscarinic acetylcholine receptor M1 | Tiotropium | 5cxv |