| Index | Gene Name | Protein Name | Drugs | PDB Code |
| 1 | CP2R1 | Vitamin D 25-hydroxylase | Cholecalciferol,Doxercalciferol,Ergocalciferol | 3c6g, 3dl9, 3czh |
| 2 | CP3A4 | Cytochrome P450 3A4 | Fluconazole,Metyrapone,Ketoconazole,Bromocriptine,Progesterone,Midazolam | 6ma7, 6ma6, 2v0m, 5vcg, 3ua1, 5a1r, 5a1p, 1w0f, 1w0g, 5te8 |
| 3 | CP2C8 | Cytochrome P450 2C8 | Montelukast,Alitretinoin,Felodipine | 2nni, 2nnh, 2nnj |
| 4 | CP51A | Lanosterol 14-alpha demethylase | Ketoconazole,Econazole,Miconazole,Isoconazole | 3ld6, 3jus |
| 5 | CP11A | Cholesterol side-chain cleavage enzyme, mitochondrial | Cholesterol | 3n9y |
| 6 | CP1A1 | Cytochrome P450 1A1 | Erlotinib | 6dwn |
| 7 | CP17A | Steroid 17-alpha-hydroxylase/17,20 lyase | Abiraterone,Pregnenolone,Progesterone | 3ruk, 4nkv, 4nkw, 4nkx |
| 8 | CP21A | Steroid 21-hydroxylase | Progesterone | 4y8w |
| 9 | CP19A | Aromatase | Testosterone | 5jkw |
| 10 | CP46A | Cholesterol 24-hydroxylase | Voriconazole,Fluvoxamine | 3mdt, 4enh |
| 11 | CP2D6 | Cytochrome P450 2D6 | Quinine | 4wnv |
| 12 | CP2C9 | Cytochrome P450 2C9 | Losartan,Warfarin | 5x24, 1og5 |
| 13 | CP2E1 | Cytochrome P450 2E1 | Pilocarpine | 3t3z |
| 14 | CP2AD | Cytochrome P450 2A13 | Pilocarpine | 3t3s |
| 15 | CP2A6 | Cytochrome P450 2A6 | Pilocarpine | 3t3r, 3t3q |
| 16 | PTGIS | Prostacyclin synthase | Minoxidil | 3b6h |