| Index | Ligand Name | Structure | PDB code | ligand desolvation |
| 1 | tn4 | Human methionine aminopeptidase type 1b (F309M mutant) in complex with TNP470 | 5yr4 | 85.9 |
| 2 | tn4 | Human methionine aminopeptidase type 1b (F309L mutant) in complex with TNP470 | 5yr6 | 84.64 |
| 3 | hm2 | Crystal structure of truncated (delta 1-89) human methionine aminopeptidase Type 1 in complex with Pyridyl pyrimidine derivative | 2g6p | 80.97 |
| 4 | yz6 | Human MetAP1 with bengamide analog YZ6, in Mn form | 4fll | 78.33 |
| 5 | tfv | Crystal structure of truncated (delta 1-89) human methionine aminopeptidase Type 1 in complex with N1-(5-chloro-6-methyl-2-(pyridin-2-yl)pyrimidin-4-yl)-N2-(5-(trifluoromethyl)pyridin-2-yl)ethane-1,2-diamine | 4ikt | 73.92 |
| 6 | hm5 | Crystal structure of type 1 human methionine aminopeptidase in complex with 3-(2,2-Dimethylpropionylamino)pyridine-2-carboxylic acid thiazole-2-ylamide | 2nq7 | 73.2 |
| 7 | shx | Crystal structure of truncated (delta 1-89) human methionine aminopeptidase Type 1 in complex with 2-((5-chloro-6-methyl-2-(pyridin-2-yl)pyrimidin-4-yl)amino)-3-phenylpropanamide | 4iku | 71.26 |
| 8 | pvp | Crystal structure of Type 1 human methionine aminopeptidase in complex with 2-(4-(5-chloro-6-methyl-2-(pyridin-2-yl)pyrimidin-4-yl)piperazin-1-yl)ethanol | 4ikr | 66.18 |
| 9 | 1ay | Pyridinylpyrimidines selectively inhibit human methionine aminopeptidase-1 | 4hxx | 64.82 |
| 10 | tfd | Crystal structure of truncated (delta 1-89) human methionine aminopeptidase Type 1 in complex with N1-(5-chloro-6-methyl-2-(pyridin-2-yl)pyrimidin-4-yl)-N2-(6-(trifluoromethyl)pyridin-2-yl)ethane-1,2-diamine | 4iks | 63.13 |