| Index | Ligand Name | Structure | PDB code | ligand desolvation |
| 1 | hzw | CRYSTAL STRUCTURE OF HUMAN METHIONINE AMINOPEPTIDASE-2 IN COMPLEX WITH AN INHIBITOR (S)-3-Hydroxy-2-oxo-1-phenyl-pyrrolidine-3-carboxylic acid 3-chloro-5-fluoro-benzylamide | 6qef | 92.72 |
| 2 | k4k | CRYSTAL STRUCTURE OF HUMAN METHIONINE AMINOPEPTIDASE-2 IN COMPLEX WITH AN INHIBITOR 2-Oxo-1-phenyl-pyrrolidine-3-carboxylic acid (2-thiophen-2-yl-ethyl)-amide | 6qeg | 91.54 |
| 3 | f77 | h-MetAP2 complexed with A773812 | 2ea2 | 90.55 |
| 4 | f79 | h-MetAP2 complexed with A797859 | 2ea4 | 90.14 |
| 5 | i96 | Human Methionine Aminopeptidase-2 Complexed with SB-587094 | 2oaz | 90.01 |
| 6 | ao2 | Crystal Structure of MetAP2 complexed with A320282 | 1r5h | 88.29 |
| 7 | hzt | CRYSTAL STRUCTURE OF HUMAN METHIONINE AMINOPEPTIDASE-2 IN COMPLEX WITH AN INHIBITOR Thiophene-2-sulfonic acid (4-fluoro-benzyl)-(4H-[1,2,4]triazol-3-ylmethyl)-amide | 6qej | 87.17 |
| 8 | hzk | CRYSTAL STRUCTURE OF HUMAN METHIONINE AMINOPEPTIDASE-2 IN COMPLEX; WITH AN INHIBITOR (S)-3-Hydroxy-2-oxo-1-(2-oxo-1,2,3,4-tetrahydro-quinolin-6-yl)-pyrrolidine-3-carboxylic acid 3-chloro-5-fluoro-benzylamide | 6qed | 85.59 |
| 9 | ao1 | Crystal Structure of MetAP2 complexed with A311263 | 1r5g | 85.21 |
| 10 | 94a | Structure of human methionine aminopeptidase 2 with covalent spiroepoxytriazole inhibitor (-)-31b | 5d6e | 82.97 |
| 11 | 52t | Structure of human methionine aminopeptidase-2 complexed with spiroepoxytriazole inhibitor (+)-31a | 5cls | 81.69 |
| 12 | a84 | h-MetAP2 complexed with A849519 | 1yw9 | 81.36 |
| 13 | tn4 | HUMAN METHIONINE AMINOPEPTIDASE 2 COMPLEXED WITH TNP-470 | 1b6a | 79.89 |
| 14 | 57r | Structure of human methionine aminopeptidase-2 complexed with spiroepoxytriazole inhibitor (+)-31b | 5d6f | 78.48 |
| 15 | ao5 | Crystal Structure of MetAP2 complexed with A357300 | 1r58 | 76.89 |
| 16 | 6ko | Potent, Reversible MetAP2 Inhibitors via FBDD | 5jhu | 75.81 |
| 17 | 7bh | CRYSTAL STRUCTURE OF HUMAN METHIONINE AMINOPEPTIDASE-2 IN COMPLEX; WITH AN INHIBITOR 6-((R)-2-o-Tolyloxymethyl-pyrrolidin-1-yl)-9H-purine | 5lyw | 75.48 |
| 18 | fug | HUMAN METHIONINE AMINOPEPTIDASE 2 COMPLEXED WITH ANGIOGENESIS INHIBITOR FUMAGILLIN | 1boa | 75.15 |
| 19 | 7bf | CRYSTAL STRUCTURE OF HUMAN METHIONINE AMINOPEPTIDASE-2 IN COMPLEX; WITH AN INHIBITOR 5-((R)-1-[1,2,4]Triazolo[1,5-a]pyrimidin-7-yl-pyrrolidin-2-ylmethoxy)-isoquinoline | 5lyx | 71.54 |
| 20 | hze | CRYSTAL STRUCTURE OF HUMAN METHIONINE AMINOPEPTIDASE-2 IN COMPLEX WITH AN INHIBITOR 5,6-Difluoro-3-(2-isopropoxy-4-piperazin-1-yl-phenyl)-1H-indole-2-carboxylic acid amide | 6qei | 68.23 |