| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | axi | The crystal structure of human abl1 T315I gatekeeper mutant kinase domain in complex with axitinib | 4twp | 0.1 |
| 2 | db8 | Structural and spectroscopic analysis of the kinase inhibitor bosutinib binding to the Abl tyrosine kinase domain | 3ue4 | 1.1 |
| 3 | 0li | AP24534, a Pan-BCR-ABL Inhibitor for Chronic Myeloid Leukemia, Potently Inhibits the T315I Mutant and Overcomes Mutation-Based Resistance | 3ik3 | 2 |
| 4 | axi | The crystal structure of human abl1 wild type kinase domain in complex with axitinib | 4wa9 | 3.8 |
| 5 | 627 | Crystal structure of the T315I Abl mutant in complex with the inhibitor PHA-739358 | 2v7a | 5 |
| 6 | 7mp | Crystal Structure of Inactive Conformation Abl Kinase Catalytic Domain Complexed with Type II Inhibitor | 2hiw | 8 |
| 7 | 0li | Crystal structure of ABL kinase domain bound with a DFG-out inhibitor AP24534 | 3oxz | 8.6 |
| 8 | p3y | Crystal Structure of the T315I Mutant of Abl kinase bound with PPY-A | 2z60 | 9 |
| 9 | 406 | Crystal structure of the c-Abl kinase domain in complex with INNO-406 | 2e2b | 11 |
| 10 | 4b7 | C-Helix-Out Binding of Dasatinib Analog to c-Abl Kinase | 4yc8 | 14 |
| 11 | p3y | Crystal Structure of Abl kinase bound with PPY-A | 2qoh | 20 |
| 12 | b91 | Structural analysis of DFG-in and DFG-out dual Src-Abl inhibitors sharing a common vinyl purine template | 3kfa | 25 |
| 13 | xy3 | Crystal structure of ABL T315I mutant kinase domain bound with a DFG-out inhibitor AP24589 | 3oy3 | 35.8 |
| 14 | 9dp | The crystal structure of human abl1 kinase domain in complex with DP-987 | 3qrk | 57 |
| 15 | jin | Abl kinase domain in complex with PD180970 | 2hzi | 70 |
| 16 | sti | CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH STI-571. | 1iep | 100 |
| 17 | 3yy | Discovery and Characterization of a Cell-Permeable, Small-molecule c-Abl Kinase Activator that Binds to the Myristoyl Binding Site | 3pyy | 137 |
| 18 | sti | Human Abl kinase domain in complex with imatinib (STI571, Glivec) | 2hyy | 170 |
| 19 | gin | Abl kinase domain in complex with NVP-AEG082 | 2hz0 | 330 |
| 20 | vx6 | Structure of the Kinase Domain of an Imatinib-Resistant Abl Mutant in Complex with the Aurora Kinase Inhibitor VX-680 | 2f4j | 2200 |