| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 1n1 | Fragment-based discovery of potent and selective DDR1/2 inhibitors | 5bvw | 1.5 |
| 2 | 4vd | Fragment-based discovery of potent and selective DDR1/2 inhibitors | 5bvn | 1.5 |
| 3 | sti | Crystal structure of the human DDR1 kinase domain in complex with imatinib | 4bkj | 1.9 |
| 4 | 4ve | Fragment-based discovery of potent and selective DDR1/2 inhibitors | 5bvo | 5 |
| 5 | di1 | Crystal structure of the human DDR1 kinase domain in complex with DDR1-IN-1 | 4ckr | 105 |
| 6 | 5wr | Structure of DDR1 receptor tyrosine kinase in complex with D2099 inhibitor at 2.25 Angstroms resolution. | 5fdp | 309 |
| 7 | 4vc | Fragment-based discovery of potent and selective DDR1/2 inhibitors | 5bvk | 1e+005 |