| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | lgv | Crystal structure of insulin-like growth factor 1 receptor (IGF-1R-WT) complex with a carbon-linked proline isostere inhibitor (34) | 3nw7 | 5.3 |
| 2 | lgw | Crystal structure of insulin-like growth factor 1 receptor (IGF-1R-WT) complex with a carbon-linked proline isostere inhibitor (11A) | 3nw6 | 7 |
| 3 | ebi | Crystal structure of insulin-like growth factor 1 receptor (IGF-1R-WT) complex with BMS-754807 [1-(4-((5-cyclopropyl-1H-pyrazol-3-yl)amino)pyrrolo[2,1-f][1,2,4]triazin-2-yl)-N-(6-fluoro-3-pyridinyl)-2-methyl-L-prolinamide] | 3i81 | 13 |
| 4 | 66a | Structure of NVP-AEW541 in complex with IGF-1R kinase | 5hzn | 61 |
| 5 | 741 | Complex Structure of Insulin-like Growth Factor Receptor and 3-Cyanoquinoline Inhibitor | 3f5p | 140 |
| 6 | d94 | Crystal structure of the insulin-like growth factor-1 receptor kinase in complex with PQIP | 3d94 | 157 |
| 7 | bmi | Structure of IGF-1R kinase domain complexed with a benzimidazole inhibitor | 2oj9 | 390 |
| 8 | 575 | Complex Structure of Insulin-like Growth Factor Receptor and Isoquinolinedione Inhibitor | 2zm3 | 614 |
| 9 | dyk | Human IGF in complex with a Dyrk1B inhibitor | 4d2r | 3300 |
| 10 | lgx | Crystal structure of insulin-like growth factor 1 receptor (IGF-1R-WT) complex with a carbon-linked proline isostere inhibitor (11B) | 3nw5 | 8400 |