The Ligandable Human Proteome

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Serine/threonine-protein kinase 24

Protein kinase domain

IndexLigand NameStructurePDB codeCompound Potency nM
1db8MST3 in complex with BOSUTINIB4qmn3
2h1nMST3 in complex with HESPERADIN4qmt10
3dkiMST3 IN COMPLEX WITH CDK1/2 INHIBITOR III, 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE4qmp14
434wMST3 IN COMPLEX WITH PF-03814735, N-{2-[(1S,4R)-6-{[4-(CYCLOBUTYLAMINO)-5-(TRIFLUOROMETHYL)PYRIMIDIN-2-YL]AMINO}-1,2,3,4-TETRAHYDRO-1,4-EPIMINONAPHTHALEN-9-YL]-2-OXOETHYL}ACETAMIDE4qmv23
5ks1MST3 IN COMPLEX WITH PP-121, 1-CYCLOPENTYL-3-(1H-PYRROLO[2,3-B]PYRIDIN-5-YL)-1H-PYRAZOLO[3,4-D]PYRIMIDIN-4-AMINE4qmw86
6627MST3 IN COMPLEX WITH Danusertib4qo9160
7b49MST3 IN COMPLEX WITH SUNITINIB4qmz210
834uMST3 in complex with CP-6734514qmq260
935rMST3 IN COMPLEX WITH AT-9283, 4-[(2-{4-[(CYCLOPROPYLCARBAMOYL)AMINO]-1H-PYRAZOL-3-YL}-1H-BENZIMIDAZOL-6-YL)METHYL]MORPHOLIN-4-IUM4qmm460
10skeMST3 IN COMPLEX WITH JNJ-7706621, 4-({5-AMINO-1-[(2,6-DIFLUOROPHENYL)CARBONYL]-1H-1,2,4-TRIAZOL-3-YL}AMINO)BENZENESULFONAMIDE4qmu1300
111n1MST3 in complex with DASATINIB4qms7400
12h8hMST3 in complex with SARACATINIB4qmx1.1e+004