| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | av9 | CRYSTAL STRUCTURE OF VEGFR2 (JUXTAMEMBRANE AND KINASE DOMAINS) IN COMPLEX WITH TIVOZANIB (AV-951) | 4ase | 0.01 |
| 2 | 900 | Crystal structure of the VEGFR2 kinase domain in complex with a naphthamide inhibitor | 3b8q | 0.5 |
| 3 | bax | Crystal Structure of VEGFR2 (Juxtamembrane and Kinase Domains) in Complex with SORAFENIB (BAY 43-9006) | 4asd | 0.52 |
| 4 | 887 | Crystal structure of the VEGFR2 kinase domain in complex with a naphthamide inhibitor | 3b8r | 0.6 |
| 5 | axi | CRYSTAL STRUCTURE OF THE VEGFR2 KINASE DOMAIN IN COMPLEX WITH AXITINIB (AG-013736) (N-Methyl-2-(3-((E)-2-pyridin-2-yl-vinyl)-1H- indazol-6-ylsulfanyl)-benzamide) | 4ag8 | 1.1 |
| 6 | 5t2 | Human Vascular Endothelial Growth Factor Receptor 2 (KDR) Kinase Domain in complex with AAL993 | 5ew3 | 1.2 |
| 7 | 0kf | Crystal Structure of the Kinase domain of Human VEGFR2 with imidazo[1,2-b]pyridazine derivative | 3vo3 | 1.4 |
| 8 | raj | Crystal structure of the VEGFR2 kinase domain in complex with a benzamide inhibitor | 3be2 | 2 |
| 9 | 0ja | Crystal Structure of the Kinase domain of Human VEGFR2 with a [1,3]thiazolo[5,4-b]pyridine derivative | 3vnt | 2.2 |
| 10 | 857 | Crystal structure of the VEGFR2 kinase domain in complex with a benzoxazole inhibitor | 2qu6 | 3 |
| 11 | gig | Crystal structure of Vegfr2 with a benzimidazole-urea inhibitor | 2oh4 | 3.5 |
| 12 | b49 | CRYSTAL STRUCTURE OF VEGFR2 (JUXTAMEMBRANE AND KINASE DOMAINS) IN COMPLEX WITH SUNITINIB (SU11248) (N-2-diethylaminoethyl)-5-((Z)-(5- fluoro-2-oxo-1H-indol-3-ylidene)methyl)-2,4-dimethyl-1H-pyrrole-3- carboxamide) | 4agd | 3.9 |
| 13 | 2rl | Crystal structure of the VEGFR2 kinase domain in complex with a 2,3-dihydro-1,4-benzoxazine inhibitor | 2rl5 | 4 |
| 14 | 03x | Crystal structure of the VEGFR2 kinase domain in complex with a pyrazolone inhibitor | 3u6j | 6.2 |
| 15 | 42q | Crystal structure of human VEGFR2 kinase domain with a novel pyrrolopyrimidine inhibitor. | 3vhe | 6.2 |
| 16 | sav | Crystal structure of VEGFR2 in complex with a 3,4,5-trimethoxy aniline containing pyrimidine | 3cjf | 6.3 |
| 17 | 276 | Crystal structure of the VEGFR2 kinase domain in complex with a benzimidazole inhibitor | 2qu5 | 8.7 |
| 18 | xin | Structure of VEGFR2 kinase domain in complex with BIBF1120 | 3c7q | 21 |
| 19 | aax | Crystal structure of VEGFR2 in complex with a 2-anilino-5-aryl-oxazole inhibitor | 1y6b | 38 |
| 20 | 608 | Crystal structure of the VEGFR2 kinase domain in complex with a nicotinamide inhibitor | 2p2i | 38 |
| 21 | 994 | Crystal structure of the VEGFR2 kinase domain in complex with a pyridinyl-triazine inhibitor | 2p2h | 68 |
| 22 | k11 | Crystal structure of the VEGFR2 kinase domain in complex with a pyridyl-pyrimidine benzimidazole inhibitor | 3ewh | 69 |
| 23 | c92 | Crystal structure of the VEGFR2 kinase domain in complex with a bisamide inhibitor | 3cpb | 2.5e+004 |