| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | 5ny | Development of a novel tricyclic class of potent and selective FIXa inhibitors | 5egm | 2.4 |
| 2 | 4m1 | Development of a novel class of potent and selective FIXa inhibitors | 4zae | 3.6 |
| 3 | 7gq | Discovery of novel aminobenzisoxazole derivatives as orally available factor IXa inhibitors | 5tnt | 4.9 |
| 4 | izx | Selective Benzothiophine Inhibitors of Factor IXa | 3lc5 | 270 |
| 5 | 4ln | Rapid development of two Factor IXa inhibitors from Hit to Lead | 4z0k | 462 |
| 6 | 4k6 | Rapid development of two Factor IXa inhibitors from Hit to Lead | 4yzu | 9000 |