The Ligandable Human Proteome

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Poly(ADP-ribose) polymerase, catalytic domain

IndexProtein NameGene Name PrimaryGene Name SynonymUniprot IDMost Potent Compound in PDB nM
1Poly [ADP-ribose] polymerase tankyrase-1 TNKS1PARP5A PARPL TIN1 TINF1 TNKS1O952710.1
2Poly [ADP-ribose] polymerase tankyrase-2 TNKS2PARP5B TANK2 TNKLQ9H2K20.5
3Poly [ADP-ribose] polymerase 1 PARP1ADPRT PPOLP098741.1
4Protein mono-ADP-ribosyltransferase PARP3 PARP3ADPRT3 ADPRTL3Q9Y6F170
5Protein mono-ADP-ribosyltransferase PARP14 PAR14BAL2 KIAA1268Q460N576
6Protein mono-ADP-ribosyltransferase PARP10 PAR10Q53GL71900