The Ligandable Human Proteome

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Protein mono-ADP-ribosyltransferase PARP3

Poly(ADP-ribose) polymerase, catalytic domain

IndexLigand NameStructurePDB codeCompound Potency nM
1ku8Human poly(ADP-ribose) polymerase 3, catalytic fragment in complex with an inhibitor KU00589483c4970
21vaHuman artd3 (parp3) - catalytic domain in complex with inhibitor ME03684l7l1000
31vcHuman artd3 (parp3) - catalytic domain in complex with inhibitor ME03984l7u2200
4m00Human artd3 (parp3) - catalytic domain in complex with inhibitor ME04004l7r9600
51vbHuman artd3 (parp3) - catalytic domain in complex with inhibitor STO15424l7n1.44e+004