The Ligandable Human Proteome

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Focal adhesion kinase 1

Protein kinase domain

IndexLigand NameStructurePDB codeligand desolvation
1yamCrystal Structure Analysis of Focal Adhesion Kinase with a Methanesulfonamide Diaminopyrimidine Inhibitor3bz387.35
24guFocal adhesion kinase catalytic domain in complex with (2-Fluoro-phenyl)-(1H-pyrazolo[3,4-d]pyrimidin-4-yl)-amine4gu985.44
3kaoFOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH 1-(5-tert-Butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-(4-pyridin-3- yl-phenyl)-urea4kao84.81
410nFOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH N-{3-[(5-Cyano-2-phenyl-1H-pyrrolo[2,3-b]pyridin-4-ylamino)- methyl]-pyridin-2-yl}-N-methyl-methanesulfonamide4gu683.4
55riFocal Adhesion Kinase catalytic domain in complex with a diarylamino- 1,3,5-triazine inhibitor4c7t81.39
6bijFocal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor2jko79.29
7bi9Focal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor2jkk78.5
8kgwFocal Adhesion Kinase catalytic domain in complex with a diarylamino- 1,3,5-triazine inhibitor4brx76.5
9biiFocal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor2jkm74.97
107pyCrystal Structure of Focal Adhesion Kinase Domain Complexed with 7H-Pyrrolo [2,3-d] pyrimidine Derivative2etm74.55
11h82Crystal structure of PTK2 in complex with BI-4464.6i8z74.04
12vg8Focal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor2jkq73.67
13euqFocal Adhesion Kinase catalytic domain in complex with irreversible inhibitor6gcw72.86
14euwFocal Adhesion Kinase catalytic domain in complex with irreversible inhibitor6gcr71.44
151bqStructure of Focal Adhesion Kinase catalytic domain in complex with hinge binding pyrazolobenzothiazine compound.4i4e70.53
16euwFocal Adhesion Kinase catalytic domain in complex with irreversible inhibitor6gcx70.42