| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | i0g | Benzopyrans are Selective Estrogen Receptor beta Agonists (SERBAs) with Novel Activity in Models of Benign Prostatic Hyperplasia | 2i0g | 0.19 |
| 2 | jj3 | Estrogen receptor beta ligand binding domain in complex with a Benzopyran agonist | 2jj3 | 0.28 |
| 3 | dc8 | Estrogen receptor beta ligand-binding domain complexed to a benzopyran ligand | 2z4b | 0.44 |
| 4 | 3as | Estrogen receptor beta ligand-binding domain complexed to a benzopyran ligand | 2qtu | 0.53 |
| 5 | fbr | Human estrogen receptor beta ligand-binding domain in complex with compound 45 | 2giu | 1.5 |
| 6 | est | STRUCTURE OF ESTRADIOL-BOUND ESTROGEN RECEPTOR BETA LBD IN COMPLEX WITH LXXLL MOTIF FROM NCOA5 | 2j7x | 1.7 |
| 7 | mon | Estrogen Receptor beta with Selective Triazine Modulator | 1nde | 15 |
| 8 | 789 | Crystal structure of estrogen receptor beta complexed with 3-Bromo-6-hydroxy-2-(4-hydroxy-phenyl)-inden-1-one | 1zaf | 20 |