| Index | Ligand Name | Structure | PDB code | Compound Potency nM |
| 1 | lsj | Crystal Structure of the Glucocorticoid Receptor Ligand Binding Domain Bound to a Dibenzoxapine Sulfonamide | 4lsj | 0.268 |
| 2 | mof | Crystal Structure of mometasone furoate-bound glucocorticoid receptor ligand binding domain | 4p6w | 0.7 |
| 3 | nn7 | The discovery of potent selective glucocorticoid receptor modulators, suitable for inhalation | 4csj | 4.9 |
| 4 | jzs | Glucocorticoid Receptor with Bound alaninamide 10 with TIF2 peptide | 3k22 | 12.59 |
| 5 | dex | CRYSTAL STRUCTURE OF THE AGONIST FORM OF GLUCOCORTICOID RECEPTOR | 1p93 | 19 |
| 6 | hcy | Crystal Structure of cortisol-bound glucocorticoid receptor ligand binding domain | 4p6x | 91 |
| 7 | 486 | Crystal Structure of the Antagonist Form of Glucocorticoid Receptor | 1nhz | 840 |