The Ligandable Human Proteome

Glucocorticoid receptor

Nuclear hormone receptor, ligand-binding domain

Index	Ligand Name	Structure	PDB code	ligand desolvation
1	mof	Crystal Structure of mometasone furoate-bound glucocorticoid receptor ligand binding domain	4p6w	99.92
2	lsj	Crystal Structure of the Glucocorticoid Receptor Ligand Binding Domain Bound to a Dibenzoxapine Sulfonamide	4lsj	99.91
3	gw6	Ligand binding domain of the glucocorticoid receptor complexed with fluticazone furoate	3cld	99.84
4	dex	GR in complex with dexamethasone	4udc	99.59
5	b9t	Glucocorticoid Receptor in complex with compound 31	6el7	99.5
6	hcy	Crystal Structure of cortisol-bound glucocorticoid receptor ligand binding domain	4p6x	99.04
7	dex	CRYSTAL STRUCTURE OF THE AGONIST FORM OF GLUCOCORTICOID RECEPTOR	1p93	99
8	866	Glucocorticoid Receptor LBD bound to GSK866	3e7c	98.93
9	dex	Crystal structure of a dimer complex of the human glucocorticoid receptor ligand-binding domain bound to dexamethasone and a TIF2 coactivator motif	1m2z	98.83
10	b9q	Glucocorticoid Receptor in complex with compound 4	6el6	98.81
11	r8c	Structure guided design and discovery of Indazole ethers as highly potent, non-steroidal Glucocorticoid receptor modulators	5g5w	98.78
12	e7t	Discovery of New Selective Glucocorticoid Receptor Agonist Leads	5g3j	98.69
13	8w8	Glucocorticoid Receptor in complex with AZD5423	5nft	98.67
14	486	Crystal structure of the antagonist form of human glucocorticoid receptor	3h52	98.52
15	nn7	The discovery of potent selective glucocorticoid receptor modulators, suitable for inhalation	4csj	98.51
16	b9w	Glucocorticoid Receptor in complex with AZD9567	6el9	97.53
17	jzs	Glucocorticoid Receptor with Bound alaninamide 10 with TIF2 peptide	3k22	96.62
18	29m	Crystal Structure of the Glucocorticoid Receptor Bound to a Non-steroidal Antagonist Reveals Repositioning and Partial Disordering of Activation Function Helix 12	4mdd	94.2
19	486	Structure of the dominant negative mutant Glucocorticoid Receptor alpha (L733K/N734P) complexed with RU-486	5uc3	92.36
20	486	Crystal Structure of the Antagonist Form of Glucocorticoid Receptor	1nhz	91.2