The Ligandable Human Proteome

Peroxisome proliferator-activated receptor delta

Nuclear hormone receptor, ligand-binding domain

Index	Ligand Name	Structure	PDB code	ligand desolvation
1	7u7	Human PPARdelta ligand-binding domain in complexed with specific agonist 9	5u3y	98.69
2	7v4	Human PPARdelta ligand-binding domain in complexed with specific agonist 3	5u3s	98.68
3	7tv	Human PPARdelta ligand-binding domain in complexed with specific agonist 5	5u3u	98.63
4	7ug	Human PPARdelta ligand-binding domain in complexed with specific agonist 16	5u41	98.61
5	7v1	Human PPARdelta ligand-binding domain in complexed with specific agonist 2	5u3r	98.61
6	7u4	Human PPARdelta ligand-binding domain in complexed with specific agonist 8	5u3x	98.57
7	d32	Crystal Structure of Peroxisome Proliferator-Activated Receptor Delta (PPARd) in Complex with a Full Agonist	3gz9	98.56
8	7uy	Human PPARdelta ligand-binding domain in complexed with specific agonist 4	5u3t	98.53
9	7uj	Human PPARdelta ligand-binding domain in complexed with specific agonist 1	5u3q	98.46
10	7ty	Human PPARdelta ligand-binding domain in complexed with specific agonist 6	5u3v	98.41
11	7ua	Human PPARdelta ligand-binding domain in complexed with specific agonist 10	5u3z	98.33
12	7sm	Human PPARdelta ligand-binding domain in complexed with specific agonist 11	5u42	98.3
13	7ss	Human PPARdelta ligand-binding domain in complexed with specific agonist 12	5u43	98.15
14	7t1	Human PPARdelta ligand-binding domain in complexed with GW501516	5u46	98.15
15	gni	3,4,5-Trisubstituted Isoxazoles as Novel PPARdelta Agonists: Part2	2j14	98.1
16	7sy	Human PPARdelta ligand-binding domain in complexed with specific agonist 14	5u45	98.09
17	89l	Co-crystal structure of Inhibitor compound in complex with human PPARdelta LBD	5xmx	98.08
18	gw0	Crystal structure PPAR delta binding GW0742	3tkm	97.88
19	8rr	Human Peroxisome proliferator-activated receptor (PPAR) delta in complexed with a potent and selective agonist	5y7x	97.63
20	l41	Crystal Structure of PPAR-delta complex	3d5f	97.52
21	7u1	Human PPARdelta ligand-binding domain in complexed with specific agonist 7	5u3w	97.45
22	401	Human PPAR delta ligand binding domain in complex with a synthetic agonist TIPP401	2znq	97.4
23	9lu	Co-crystal structure of an Inhibitor in complex with human PPARdelta LBD	5zxi	97.38
24	k55	Human PPAR delta ligand binding domain in complex with a synthetic agonist TIPP204	2znp	97.06
25	il2	Structural basis for iloprost as a dual PPARalpha/delta agonist	3sp9	97.01
26	z00	Novel Sulfonylthiadiazoles with an Unusual Binding Mode as Partial Dual Peroxisome Proliferator-Activated Receptor (PPAR) gamma-delta Agonists with High Potency and In-vivo Efficacy	2xyx	96.54
27	dy6	PPARdelta complexed with an anthranilic acid partial agonist	3dy6	96.53
28	7sv	Human PPARdelta ligand-binding domain in complexed with specific agonist 13	5u44	96.33
29	3oz	PPAR Delta in complex with azppard02	3oz0	95.94
30	433	MOLECULAR RECOGNITION OF FATTY ACIDS BY PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS	1gwx	94.27
31	331	Crystal structure of PPAR delta complexed with GW2331	1y0s	93.91
32	1fa	Ligand binding domain of PPAR delta receptor in complex with a partial agonist	2q5g	89.38